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  Synthesis and analytical applications of sodium N-bromo-p-nitrobenzenesulfonamide

  Made Gowda, N. M., Trieff, N. M., Sadagopa Ramanujam, V. M., Malinski, T., Kadish, K. M. & Mahadevappa, D. S., 1983, In: Analytica Chimica Acta. 147, C, p. 429-433 5 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis and anticancer activity of novel oleanolic acid derivatives

  Ding, Y., Zhang, Z. Z., Huang, Z. J., Mou, Y., Ji, H., Lai, Y. S. & Zhang, Y. H., Oct 1 2011, In: Journal of China Pharmaceutical University. 42, 5, p. 385-391 7 p.

  Research output: Contribution to journal › Article › peer-review
  4 Scopus citations

• Synthesis and antitumor activity of NO-donating CDDO analogues

  Zhang, S. B., Zhang, Z. Z., Ding, Y., Lai, Y. S., Mou, Y., Ai, Y., Ji, H. & Zhang, Y. H., Aug 1 2012, In: Journal of China Pharmaceutical University. 43, 4, p. 293-297 5 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis and antiviral activity of 4,6-disubstituted pyrimido[4,5-b]indole ribonucleosides

  Tichý, M., Pohl, R., Xu, H. Y., Chen, Y. L., Yokokawa, F., Shi, P. Y. & Hocek, M., Oct 15 2012, In: Bioorganic and Medicinal Chemistry. 20, 20, p. 6123-6133 11 p.

  Research output: Contribution to journal › Article › peer-review
  43 Scopus citations

• Synthesis and Biochemical Evaluation of Noncyclic Nucleotide Exchange Proteins Directly Activated by cAMP 1 (EPAC1) Regulators

  Wang, P., Luchowska-Stańska, U., Van Basten, B., Chen, H., Liu, Z., Wiejak, J., Whelan, P., Morgan, D., Lochhead, E., Barker, G., Rehmann, H., Yarwood, S. J. & Zhou, J., May 28 2020, In: Journal of medicinal chemistry. 63, 10, p. 5159-5184 26 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis and biological activity of new 6- and 7-substituted 2β- butyl-3-phenyltropanes as ligands for the dopamine transporter

  Prakash, K. R. C., Araldi, G. L., Smith, M. P., Zhang, M., Johnson, K. M. & Kozikowski, A. P., Jan 1 1998, In: Medicinal Chemistry Research. 8, 1-2, p. 43-58 16 p.

  Research output: Contribution to journal › Article › peer-review
  3 Scopus citations

• Synthesis and biological evaluation of 1-azabicyclo-[3.2.1]octanes: New dopamine transporter inhibitors

  Tamiz, A. P., Smith, M. P., Enyedy, I., Flippen-Anderson, J., Zhang, M., Johnson, K. M. & Kozikowski, A. P., Aug 7 2000, In: Bioorganic and Medicinal Chemistry Letters. 10, 15, p. 1681-1686 6 p.

  Research output: Contribution to journal › Article › peer-review
  4 Scopus citations

• Synthesis and biological evaluation of new bisindole-imidazopyridine hybrids as apoptosis inducers

  Sunkari, S., Bonam, S. R., Rao, A. V. S., Riyaz, S., Lakshma Nayak, V., Kumar, H. M. S., Kamal, A. & Nagendra Babu, B., Jun 2019, In: Bioorganic Chemistry. 87, p. 484-494 11 p.

  Research output: Contribution to journal › Article › peer-review
  11 Scopus citations

• Synthesis and biological evaluation of oxadiazole derivatives as inhibitors of soluble guanylyl cyclase

  von Wantoch Rekowski, M., Pyriochou, A., Papapetropoulos, N., Stößel, A., Papapetropoulos, A. & Giannis, A., Feb 1 2010, In: Bioorganic and Medicinal Chemistry. 18, 3, p. 1288-1296 9 p.

  Research output: Contribution to journal › Article › peer-review
  21 Scopus citations

• Synthesis and biological evaluation of two novel DAT-binding technetium complexes containing a piperidine based analogue of cocaine

  Hoepping, A., Babich, J., Zubieta, J. A., Johnson, K. M., Machill, S. & Kozikowski, A. P., Nov 15 1999, In: Bioorganic and Medicinal Chemistry Letters. 9, 22, p. 3211-3216 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  15 Scopus citations

• Synthesis and biological properties of new 2β-alkyl- and 2β-aryl-3- (substituted phenyl)tropane derivatives: Stereochemical effect of C-3 on affinity and selectivity for neuronal dopamine and serotonin transporters

  Kozikowski, A. P., Araldi, G. L., Prakash, K. R. C., Zhang, M. & Johnson, K. M., Dec 3 1998, In: Journal of medicinal chemistry. 41, 25, p. 4973-4982 10 p.

  Research output: Contribution to journal › Article › peer-review
  24 Scopus citations

• Synthesis and characterization of isotopically enriched pyrimidine deoxynucleoside oxidation damage products

  LaFrancois, C. J., Fujimoto, J. & Sowers, L. C., 1998, In: Chemical Research in Toxicology. 11, 1, p. 75-83 9 p.

  Research output: Contribution to journal › Article › peer-review
  47 Scopus citations

• Synthesis and characterization of oligonucleotides containing 5-chlorocytosine

  Kang, J. I., Burdzy, A., Liu, P. & Sowers, L. C., Sep 2004, In: Chemical Research in Toxicology. 17, 9, p. 1236-1244 9 p.

  Research output: Contribution to journal › Article › peer-review
  24 Scopus citations

• Synthesis and cleavage of oligodeoxynucleotides containing a 5- hydroxyuracil residue at a defined site

  Fujimoto, J., Tran, L. & Sowers, L. C., 1997, In: Chemical Research in Toxicology. 10, 11, p. 1254-1258 5 p.

  Research output: Contribution to journal › Article › peer-review
  29 Scopus citations

• Synthesis and c-met kinase inhibition of 3,5-disubstituted and 3,5,7-trisubstituted quinolines: Identification of 3-(4-acetylpiperazin-1-yl)-5- (3-nitrobenzylamino)-7- (trifluoromethyl)quinoline as a novel anticancer agent

  Wang, Y., Ai, J., Wang, Y., Chen, Y., Wang, L., Liu, G., Geng, M. & Zhang, A., Apr 14 2011, In: Journal of medicinal chemistry. 54, 7, p. 2127-2142 16 p.

  Research output: Contribution to journal › Article › peer-review
  56 Scopus citations

• Synthesis and Crystal Structure of 1-(o-methylphenyl)-2- (p-methoxyphenyl)-1,3,2-diazaphospholidin-4-thione-2-sulfide

  He, L. N., Chen, R. Y., Zhou, J., Hong-Gen, W. & Xin-Kan, Y., 1997, In: Jiegou Huaxue. 16, 3, p. 215-218 4 p.

  Research output: Contribution to journal › Article › peer-review
  7 Scopus citations

• Synthesis and crystal structure of 2-phosphonoalkyl-1, 2-benzisoselenazol-3(2H)-ones and their antitumor activities

  Zhou, J. & Chen, R., Jan 1 1999, In: Heteroatom Chemistry. 10, 3, p. 247-254 8 p.

  Research output: Contribution to journal › Article › peer-review
  10 Scopus citations

• Synthesis and crystal structure of α-(3-phenylureido)-α-(2,4-dichloroptienyl) methyl phenylphosphinic acid

  Zhou, J., Chen, R. Y., Wang, H. G. & Yao, X. K., Dec 1 1997, In: Jiegou Huaxue. 16, 3, p. 207-210 4 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis and evaluation of dimeric derivatives of 5-HT _2A receptor (5-HT _2AR) antagonist M-100907

  Shashack, M. J., Cunningham, K. A., Seitz, P. K., McGinnis, A., Smith, T. D., Watson, C. & Gilbertson, S. R., Nov 16 2011, In: ACS chemical neuroscience. 2, 11, p. 640-644 5 p.

  Research output: Contribution to journal › Article › peer-review
  16 Scopus citations

• Synthesis and evaluation of iodine-123 labelled tricyclic tropanes as radioligands for the serotonin transporter

  Quinlivan, M., Mattner, F., Papazian, V., Zhou, J., Katsifis, A., Emond, P., Chalon, S., Kozikowski, A., Guilloteau, D. & Kassiou, M., Oct 2003, In: Nuclear Medicine and Biology. 30, 7, p. 741-746 6 p.

  Research output: Contribution to journal › Article › peer-review
  10 Scopus citations

• Synthesis and Herbicidal Activity of 1-Aryl-2-phenyI-3-methyl-3-isopropyl-1,4,2-diazaphospholidin-5-one-2-oxides

  Zhou, J., Qiu, Y. G., Feng, K. S. & Chen, R. Y., Jul 10 1999, In: Kao Teng Hsueh Hsiao Hua Heush Hsueh Pao/ Chemical Journal of Chinese Universities. 20, 7, 1 p.

  Research output: Contribution to journal › Article › peer-review
  3 Scopus citations

• Synthesis and in vitro efficacy studies of silver carbene complexes on biosafety level 3 bacteria

  Panzner, M. J., Deeraksa, A., Smith, A., Wright, B. D., Hindi, K. M., Kascatan-Nebioglu, A., Torres, A. G., Judy, B. M., Hovis, C. E., Hilliard, J. K., Mallett, R. J., Cope, E., Estes, D. M., Cannon, C. L., Leid, J. G. & Youngs, W. J., May 2009, In: European Journal of Inorganic Chemistry. 13 SPEC. ISS., p. 1739-1745 7 p.

  Research output: Contribution to journal › Article › peer-review
  60 Scopus citations

• Synthesis and mutagenesis of the butadiene-derived N3 2′-deoxyuridine adducts

  Fernandes, P. H., Hackfeld, L. C., Kozekov, I. D., Hodge, R. P. & Lloyd, R. S., Jul 2006, In: Chemical Research in Toxicology. 19, 7, p. 968-976 9 p.

  Research output: Contribution to journal › Article › peer-review
  12 Scopus citations

• Synthesis and pharmacological evaluation of (Z)-9-(Heteroarylmethylene)-7-azatricyclo[4.3.1.0^3,7]decanes: Thiophene analogues as potent norepinephrine transporter inhibitors

  Zhou, J., Kläß, T., Zhang, A., Johnson, K. M., Wang, C. Z., Ye, Y. & Kozikowski, A. P., Oct 20 2003, In: Bioorganic and Medicinal Chemistry Letters. 13, 20, p. 3565-3569 5 p.

  Research output: Contribution to journal › Article › peer-review
  6 Scopus citations

• Synthesis and pharmacological evaluation of non-catechol G protein biased and unbiased dopamine D1 receptor agonists

  Wang, P., Felsing, D., Chen, H., Raval, S., Allen, J. & Zhou, J., May 9 2019, In: ACS Medicinal Chemistry Letters. 10.1021/acsmedchemlett.9b00050, p. 792-799 8 p., 10.1021/acsmedchemlett.9b00050.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  11 Scopus citations

• Synthesis and Pharmacological Evaluation of Novel Adenine-Hydrogen Sulfide Slow Release Hybrids Designed as Multitarget Cardioprotective Agents

  Lougiakis, N., Papapetropoulos, A., Gikas, E., Toumpas, S., Efentakis, P., Wedmann, R., Zoga, A., Zhou, Z., Iliodromitis, E. K., Skaltsounis, A. L., Filipovic, M. R., Pouli, N., Marakos, P. & Andreadou, I., Mar 10 2016, In: Journal of medicinal chemistry. 59, 5, p. 1776-1790 15 p.

  Research output: Contribution to journal › Article › peer-review
  22 Scopus citations

• Synthesis and properties of defined DNA oligomers containing base mispairs involving 2-aminopurine

  Eritja, R., Kaplan, B. E., Mhaskar, D., Sowers, L. C., Petruska, J. & Goodman, M. F., Jul 11 1986, In: Nucleic acids research. 14, 14, p. 5869-5884 16 p.

  Research output: Contribution to journal › Article › peer-review
  20 Scopus citations

• Synthesis and properties of novel amino acid linked phosphoryl nitrogen mustard derivatives

  Chen, RY. Y., Wang, HL. L. & Zhou, J., 1994, In: Heteroatom Chemistry. 5, 5-6, p. 497-501 5 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis and properties of novel nitrogen mustard linked phosphoryl diamide derivatives

  Chen, R. Y., Mao, L. J., Wang, H. L. & Zhou, J., Apr 1 1994, In: Phosphorus, Sulfur, and Silicon and the Related Elements. 89, 1-4, p. 89-95 7 p.

  Research output: Contribution to journal › Article › peer-review
  1 Scopus citations

• Synthesis and properties of novel α-phosphoryl(thio)ureido alkanephosphonate derivatives

  Zhou, J. & Chen, R. Y., 1996, In: Phosphorus, Sulfur and Silicon and Related Elements. 118, 1-4, p. 247-256 10 p.

  Research output: Contribution to journal › Article › peer-review

• Synthesis and Rational design of Europium and Lithium Doped Sodium Zinc Molybdate with Red Emission for Optical Imaging

  Jain, N., Paroha, R., Singh, R. K., Mishra, S. K., Chaurasiya, S. K., Singh, R. A. & Singh, J., Dec 1 2019, In: Scientific reports. 9, 1, 2472.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  34 Scopus citations

• Synthesis and screening of small molecule inhibitors of anthrax edema factor

  Jimenez, M. E., Bush, K., Pawlik, J., Sower, L., Peterson, J. W. & Gilbertson, S. R., Jul 15 2008, In: Bioorganic and Medicinal Chemistry Letters. 18, 14, p. 4215-4218 4 p.

  Research output: Contribution to journal › Article › peer-review
  9 Scopus citations

• Synthesis and Secretion of Transferrin by Cultured Mouse Hepatoma Cells

  PAPACONSTANTINOU, JOHN., HILL, ROBERT. E., GIBSON, WILLIAM. H. & RAO, EDITH. Y., 1978, In: Differentiation. 10, 1-3, p. 139-145 7 p.

  Research output: Contribution to journal › Article › peer-review
  1 Scopus citations

• Synthesis and stereochemistry of new cyclic phosphate-phosphonates

  Zhou, J. & Chen, R. Y., Dec 1 1997, In: Chinese Chemical Letters. 8, 1, p. 11-12 2 p.

  Research output: Contribution to journal › Article › peer-review
  1 Scopus citations

• Synthesis and structural characterization of metal complexes based on pyrazole/imidazolium chlorides

  Lee, H. M., Chiu, P. L., Hu, C. H., Lai, C. L. & Chou, Y. C., Jan 17 2005, In: Journal of Organometallic Chemistry. 690, 2, p. 403-414 12 p.

  Research output: Contribution to journal › Article › peer-review
  84 Scopus citations

• Synthesis and structure-activity relationships of 3-[(2-methyl-1,3-thiazol- 4-yl)ethynyl]pyridine analogues as potent, noncompetitive metabotropic glutamate receptor subtype 5 antagonists; search for cocaine medications

  Iso, Y., Grajkowska, E., Wroblewski, J. T., Davis, J., Goeders, N. E., Johnson, K. M., Sanker, S., Roth, B. L., Tueckmantel, W. & Kozikowski, A. P., Feb 9 2006, In: Journal of medicinal chemistry. 49, 3, p. 1080-1100 21 p.

  Research output: Contribution to journal › Article › peer-review
  44 Scopus citations

• Synthesis and Structure-Activity Relationships of Tool Compounds Based on WAY163909, a 5-HT_2C Receptor Agonist

  Chen, Y. C., Hartley, R. M., Anastasio, N. C., Cunningham, K. A. & Gilbertson, S. R., May 17 2017, In: ACS chemical neuroscience. 8, 5, p. 1004-1010 7 p.

  Research output: Contribution to journal › Article › peer-review
  7 Scopus citations

• Synthesis and structure–activity relationship studies of MI-2 analogues as MALT1 inhibitors

  Wu, G., Wang, H., Zhou, W., Zeng, B., Mo, W., Zhu, K., Liu, R., Zhou, J., Chen, C. & Chen, H., Jul 23 2018, In: Bioorganic and Medicinal Chemistry. 26, 12, p. 3321-3344 24 p.

  Research output: Contribution to journal › Article › peer-review
  12 Scopus citations

• Synthesis and utilization of ¹³C(8)-enriched purines

  LaFrancois, C. J., Fujimoto, J. & Sowers, L. C., 1999, In: Nucleosides and Nucleotides. 18, 1, p. 23-37 15 p.

  Research output: Contribution to journal › Article › peer-review
  3 Scopus citations

• Synthesis and vectorial export of cGMP in airway epithelium: Expression of soluble and CNP-specific guanylate cyclases

  Geary, C., Goy, M. F. & Boucher, R. C., 1993, In: AM.J.PHYSIOL.. 265, 6 part 1

  Research output: Contribution to journal › Article › peer-review

• Synthesis and vectorial export of cGMP in airway epithelium: Expression of soluble and CNP-specific guanylate cyclases

  Geary, C. A., Goy, M. F. & Boucher, R. C., 1993, In: American Journal of Physiology - Lung Cellular and Molecular Physiology. 265, 6 9-6, p. L598-L605

  Research output: Contribution to journal › Article › peer-review
  11 Scopus citations

• Synthesis hydrolysis of oligodeoxyribonucleotides containing 2-aminopurine

  Fujimoto, J., Nuesca, Z., Mazurek, M. & Sowers, L. C., 1996, In: Nucleic acids research. 24, 4, p. 754-759 6 p.

  Research output: Contribution to journal › Article › peer-review

  Open Access
  30 Scopus citations

• Synthesis of 1,4-benzothiazin-2-yl derivatives of 1,3-dicarbonyl compounds and benzothiazinone spiro derivatives by the reaction of 2-chloro-1,4-benzothiazin-3-ones with 'push-pull' enamines

  Nazarenko, K. G., Shtil, N. A., Buth, S. A., Chernega, A. N., Lozinskii, M. O. & Tolmachev, A. A., May 5 2008, In: Tetrahedron. 64, 19, p. 4478-4485 8 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis of 1- and 1,2,2′-Deuteriated Deoxyribose and Incorporation into Deoxyribonucleosides

  Hodge, R. P., Brush, C. K., Harris, C. M. & Harris, T. M., Feb 1 1991, In: Journal of Organic Chemistry. 56, 4, p. 1553-1564 12 p.

  Research output: Contribution to journal › Article › peer-review
  8 Scopus citations

• Synthesis of 2-(p-toluenesulfonamido)-4-phenyl-4,5-dihydro-1H-1,3,4- diazaphosphole 4-oxides

  Zhou, J., Qiu, Y., Feng, K. & Chen, R. Y., 1998, In: Synthetic Communications. 28, 24, p. 4673-4678 6 p.

  Research output: Contribution to journal › Article › peer-review
  3 Scopus citations

• Synthesis of 3, 4-diphenyl-l, 3, 4- diazaphospholidin-2-thione-4-oxides and their quantitative structure-herbicidal activity relationship

  Wang, H. L., Zhou, J., Qiu, Y. G., Feng, K. S. & Chen, R. Y., Jul 1 1995, In: Phosphorus, Sulfur, and Silicon and the Related Elements. 104, 1-4, p. 135-141 7 p.

  Research output: Contribution to journal › Article › peer-review
  3 Scopus citations

• Synthesis of 4′-ester analogs of resveratrol and their evaluation in malignant melanoma and pancreatic cell lines

  Wong, Y., Osmond, G., Brewer, K. I., Tyler, D. S. & Andrus, M. B., Feb 1 2010, In: Bioorganic and Medicinal Chemistry Letters. 20, 3, p. 1198-1201 4 p.

  Research output: Contribution to journal › Article › peer-review
  19 Scopus citations

• Synthesis of 5-polyfluoroalkyl-4-(p-tolyl-sulfonyl)pyrazoles and 4-polyfluoroalkyl-5-(p-tolylsulfonyl)pyrimidines from 1-dimethylamino-2-(p- tolylsulfonyl)-polyfluoro-1-alken-3-ones

  Kanishchev, O. S., Bandera, Y. P., Timoshenko, V. M., Rusanov, E. B., But, S. A. & Shermolovich, Y. G., Jul 2007, In: Chemistry of Heterocyclic Compounds. 43, 7, p. 887-892 6 p.

  Research output: Contribution to journal › Article › peer-review
  14 Scopus citations

• Synthesis of 8-oxa analogues of norcocaine endowed with interesting cocaine-like activity

  Kozikowski, A. P., Simoni, D., Roberti, M., Rondanin, R., Wang, S., Du, P. & Johnson, K. M., Jul 5 1999, In: Bioorganic and Medicinal Chemistry Letters. 9, 13, p. 1831-1836 6 p.

  Research output: Contribution to journal › Article › peer-review
  15 Scopus citations

• Synthesis of a new class of glycolipids and the evaluation of their immunogenicity using murine splenocytes

  Sandeep, A., Reddy, B. S., Hyder, I. & Kumar, H. M. S., Jul 23 2016, In: Journal of Carbohydrate Chemistry. 35, 6, p. 326-343 18 p.

  Research output: Contribution to journal › Article › peer-review
  6 Scopus citations