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Discovery of 3-((4-Benzylpyridin-2-yl)amino)benzamides as Potent GPR52 G Protein-Biased Agonists
Ryan Murphy
, Pingyuan Wang
, Saghir Ali
, Hudson Smith
, Daniel Felsing
, Haiying Chen
,
Jia Zhou
,
John Allen
Pharmacology & Toxicology
Center for Addiction Sciences and Therapeutics
Research output
:
Contribution to journal
›
Article
›
peer-review
1
Scopus citations
Overview
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Dive into the research topics of 'Discovery of 3-((4-Benzylpyridin-2-yl)amino)benzamides as Potent GPR52 G Protein-Biased Agonists'. Together they form a unique fingerprint.
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Keyphrases
Amino
100%
Arrestin
14%
Benzamide
100%
Bias Potential
14%
Biased Agonism
14%
Biased Agonist
100%
Brain Exposure
14%
CAMP Signaling
14%
Desensitization
14%
Drug Design Strategies
14%
G Protein
100%
GPR52
100%
Neurological Diseases
14%
Neuropsychiatric Diseases
14%
Neurotherapeutics
14%
Parent Compounds
14%
Pharmacological Tools
14%
Signaling Bias
14%
Target Selectivity
14%
Therapeutic Potential
14%
Pharmacology, Toxicology and Pharmaceutical Science
Benzamide Derivative
100%
Desensitization
50%
Drug Development
50%
Guanine Nucleotide Binding Protein
100%
Mental Diseases
50%
Neurologic Disease
50%
Retina S Antigen
50%