Discovery of potent and selective nonplanar tankyrase inhibiting nicotinamide mimics

Yves Nkizinkiko, B. V.S. Suneel Kumar, Variam Ullas Jeankumar, Teemu Haikarainen, Jarkko Koivunen, Chanduri Madhuri, Perumal Yogeeswari, Harikanth Venkannagari, Ezeogo Obaji, Taina Pihlajaniemi, Dharmarajan Sriram, Lari Lehtiö

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Biochemistry, Genetics and Molecular Biology

Pharmacology, Toxicology and Pharmaceutical Science