Keyphrases
2-Aminopyrimidine
100%
5-HT3AR
25%
AChBP
100%
Allosteric Behavior
12%
Antagonism
12%
Aromatic Side Chains
12%
Binding Mode
12%
Binding Pose
12%
Co-agonist
12%
Co-crystallization
12%
Complementary DNA (cDNA)
12%
Cooperative Interaction
12%
Fluorescent Reporter
12%
HEK Cells
12%
Heteromer
12%
IC50 Value
12%
Kd Values
12%
Ligand Binding
12%
Ligand Complexes
12%
Ligand-gated Ion Channel
12%
Nicotinic Acetylcholine Receptor (nAChR)
100%
Nicotinic Agonists
50%
Partial Agonist
12%
Receptor Activation
100%
Receptor Subtypes
12%
Receptor-ligand Interaction
12%
Serotonin Receptors
12%
Structural Family
12%
Structural Features
12%
Subunit Interface
12%
Pharmacology, Toxicology and Pharmaceutical Science
Acetylcholine
100%
Agonist-Antagonist
14%
Binding Protein
100%
EC50
14%
Ligand Gated Ion Channel
14%
Nicotinic Agent
28%
Nicotinic Receptor
100%
Nicotinic Receptor Blocking Agent
28%
Partial Agonist
14%
Receptor
28%
Receptor Subtype
14%
Serotonin 5 Receptor
14%
Biochemistry, Genetics and Molecular Biology
5-HT Receptor
14%
Acetylcholine
100%
Agonist
42%
Binding Protein
100%
EC50
14%
Ligand Binding
14%
Ligand-Gated Ion Channel
14%
Nicotinic Acetylcholine Receptor
100%
Nicotinic Agonist
28%
Nicotinic Antagonist
28%
Chemistry
Acetylcholine
100%
Aminopyrimidine
100%
Binding Protein
100%
Co Crystallization
7%
EC50
7%
Kd
7%
Ligand Binding
7%
Nicotinic Agonist
15%
Nicotinic Antagonist
15%
Partial Agonist
7%
Serotonin
7%